LKT/VAPREOTIDE/V0160/2.5 mg-免疫在线蚂蚁淘旗下平台

商品详细LKT/VAPREOTIDE/V0160/2.5 mg

LKT/VAPREOTIDE/V0160/2.5 mg

商品编号： V0160-2.5mg

品牌： lktlabs

市场价： ¥8300.00

美元价： 4980.00

产地：美国(厂家直采)

公司：

产品分类：临床研究

公司分类： clinical_research

联系Q Q： 3392242852

电话号码： 4000-520-616

电子邮箱： info@ebiomall.com

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商品介绍

ProductIDV0160

CasNo.103222-11-3

Purity≥95%

Description
ProductInfo
ShippingandStorage
Downloads
References

Description

Vapreotideisasyntheticpeptideanalogofsomatostatinthatactivatessomatostatin2receptorsandinhibitsneurokinin1receptors.Vapreotideexhibitsanti-inflammatory,antiviral,orexigenic,antihypertensive,andanticancerchemotherapeuticactivities.Inmacrophages,vapreotideinhibitssubstanceP-inducedproductionofIL-8andMCP-1,preventingHIV-1infection.Intheclinicaltreatmentofprostatecancer,vapreotidedecreasesPSAandPAPlevelsandbonepainscores.Additionally,thiscompounddecreasesportalpressureandbloodflow,improvingbleedingcontrolandmortalityratesinclinicalsubjectswithvaricealbleeding.Vapreotidealsoincreasesfoodintakeinvivo.

ProductInfo

CasNo.	103222-11-3
Purity	≥95%
Formula	C₅₇H₇₀N₁₂O₉S₂
FormulaWt.	1131.4
ChemicalName	L-Tryptophanamide,D-phenylalanyl-L-cysteinyl-L-tyrosyl-D-tryptophyl-L-lysyl-L-valyl-L-cysteinyl-,cyclic(2->7)-
IUPACName	(4R,7S,10S,13S,16S,19R)-10-(4-aminobutyl)-N-[(2R)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide
Synonym	SanvarIR;BMY41606;RC160
Appearance	Whitetooffwhitepowder

ShippingandStorage

StoreTemp	-20°C
ShipTemp	Ambient

Downloads

InfoSheet	V0160InfoSheetPDF

References

SpitsinS,TulucF,MeshkiJ,etal.AnalogofsomatostatinvapreotideexhibitsBIOLOGicaleffectsinvitroviainteractionwithneurokinin-1receptor.Neuroimmunomodulation.2013;20(5):247-55.PMID:23921645.

TachibanaT,ClineMA,KhanMS,etal.FeedingresponsestocentraladmiNISTrationofseveralsomatostatinanalogsinchicks.CompBiochemPhysiolAMolIntegrPhysiol.2011Jan;158(1):47-51.PMID:20826222.

CalèsP.Vapreotideacetateforthetreatmentofesophagealvaricealbleeding.ExpertRevGastroenterolHepatol.2008Apr;2(2):185-92.PMID:19072353.

González-BarcenaD,SchallyAV,VADIllo-BuenfilM,etal.ResponseofpatientswithadvancedprostaticcancertoadministrationofsomatostatinanalogRC-160(vapreotide)atthetimeofrelapse.Prostate.2003Aug1;56(3):183-91.PMID:12772187.

品牌介绍

LKT Labs LKT Labs 是一家专注于防癌抗癌特殊化学品研究和开发的公司。主要提供：癌症药物、药物发现试剂盒、天然产物、广泛的生命科学研究试剂、定制合成。美国LKT Labs 是1988年在美国成立的，为全球提供先端的药物研发试剂、试剂盒、委托合成，并为药物生产企业提供原料，最近几年在农药、水产养殖业有很大程度的开发。在LKT Labs 可以找到在其他地方找不到的产品。试剂