ValdecoxibisaCOXinhibitorspecificforCOX-2;italsoinhibitscarbonicanhydrase.Valdecoxibisanon-steroidalanti-inflammatorydrug(NSAID)thatexhibitsanti-inflammatoryandanalgesicactivities.Inadditiontoitsmediationofinflammatorysignaling,valdecoxibalsoactivatescannABInoid1(CB1)receptorsinvivo,modulatingglutamatesignalingandGABArelease.Valdecoxibhasbeenremovedfromclinicaluseduetoincreasedriskofthromboticeffects.
| CasNo. | 181695-72-7 |
|---|---|
| Purity | ≥98% |
| Formula | C16H14N2O3S |
| FormulaWt. | 314.36 |
| IUPACName | 4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)benzenesulfonamide |
| MeltingPoint | 162-164℃ |
| Solubility | Water0.5mg/ml |
| Appearance | WhiteCrystalPowder |
| StoreTemp | Ambient |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | V0245InfoSheetPDF |
|---|
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