A-803467isablockerofNav1.8(SCN10A)Na+channelsthatexhibitsantinociceptiveandantiarrhythmicactivities;itmayalsoblockNav1.5(SCN5A)Na+channels.A-803467inhibitsmechanicalandthermalpainnociceptioninvivo.ThiscompoundalsoblockscardiacNa+currentsandaltersactionpotentialmorphologyinventricularmyocytes.
| CasNo. | 944261-79-4 |
|---|---|
| Purity | ≥98% |
| Formula | C19H16ClNO4 |
| FormulaWt. | 357.79 |
| IUPACName | 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)-2-furamide |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | A0001InfoSheetPDF |
|---|
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