Description
Dalcetrapibisacholesterolestertransferprotein(CETP)inhibitorthatexhibitsanti-atheroscleroticactivity.Inaclinicalsetting,dalcetrapibincreasesHDLlevelsbuthasexhibitedmixedresultsregardingcardiovasculardiseaseriskreduction.
Dalcetrapibisacholesterolestertransferprotein(CETP)inhibitorthatexhibitsanti-atheroscleroticactivity.Inaclinicalsetting,dalcetrapibincreasesHDLlevelsbuthasexhibitedmixedresultsregardingcardiovasculardiseaseriskreduction.
Purity | ≥98% |
---|---|
Formula | C23H35NO2S |
FormulaWt. | 389.60 |
Synonym | JTT-705,RO4607381 |
Appearance | WhitePowder |
StoreTemp | -20°C |
---|
InfoSheet | D0244InfoSheetPDF |
---|
SchwartzGG,OlssonAG,AbtM,etal.Effectsofdalcetrapibinpatientswitharecentacutecoronarysyndrome.NEnglJMed.2012Nov29;367(22):2089-99.PMID:23126252.
GoldbergAS,HegeleRA.Cholesterylestertransferproteininhibitorsfordyslipidemia:focusondalcetrapib.DrugDesDevelTher.2012;6:251-9.PMID:23055695.
RobinsonJG.Dalcetrapib:areviewofPhaseIIdata.ExpertOpinInvestigDrugs.2010Jun;19(6):795-805.PMID:20465364.