Cyclopiazonic acid is an inhibitor of sarco/endoplasmic reticulum Ca2+/ATPase (SERCA) pumps, increasing intracellular Ca2+ levels and altering contractility in smooth muscle tissues. Additionally, this compound inhibits proliferation of Plasmodium falciparum, exhibiting some potential anti-parasitic activity.
| Cas No. | 18172-33-3 |
|---|---|
| Purity | ≥98%, TLC |
| Formula | C20H20N2O3 |
| Formula Wt. | 336.39 |
| Solubility | DMSO, Methylene Chloride and Methanol. |
| Appearance | Off-white powder |
| Store Temp | 4°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet | C9809 Info Sheet PDF |
|---|
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Darby PJ, Kwan CY, Daniel EE. Use of calcium pump inhibitors in the study of calcium regulation in smooth muscle. Biol Signals. 1993 Sep-Oct;2(5):293-304. PMID: 8038861.
