Azaperoneisabutyrophenonetranquilizerthatexhibitssedativeactivitythroughtheinhibitionofα-adrenergicreceptors.Azaperonealsoinhibitsdopaminereceptorsandhistaminereceptors;italsomaydisplayantiemetic,antipsychotic,antihistaminergic,andanticholinergicactivities.
| CasNo. | 1649-18-9 |
|---|---|
| Purity | ≥98% |
| Formula | C19H22FN3O |
| FormulaWt. | 327.40 |
| ChemicalName | 1-(4-Fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-1-butanone |
| IUPACName | 1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one |
| Synonym | Stresnil;Suicalm |
| MeltingPoint | 73-75°C |
| Solubility | Solubleinchloroformandethylacetate. |
| Appearance | AWhiteorAlmostWhiteCrystallinePowder |
| StoreTemp | 4°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | A9801InfoSheetPDF |
|---|
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