Description
Thispeptideinhibitscalcineurinphosphataseactivityandisusedtoexaminetheeffectsofcalcineurininresearchstudies.Incellularmodels,thispeptideinhibitscalcineurin-inducedglutamate-mediatedneuronalcelldeathanddecreasesL-typeCa2+channelcurrents.
Thispeptideinhibitscalcineurinphosphataseactivityandisusedtoexaminetheeffectsofcalcineurininresearchstudies.Incellularmodels,thispeptideinhibitscalcineurin-inducedglutamate-mediatedneuronalcelldeathanddecreasesL-typeCa2+channelcurrents.
| Purity | ≥95% |
|---|---|
| Formula | C124H205N39O39S2 |
| FormulaWt. | 2930.38 |
| Appearance | Whitetooffwhitepowder |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | C0247InfoSheetPDF |
|---|
TeradaH,MatsushitaM,LuYF,etal.Inhibitionofexcitatoryneuronalcelldeathbycell-permeablecalcineurinautoinhibitorypeptide.JNeuRochem.2003Dec;87(5):1145-51.PMID:14622094.
NorrisCM,BlalockEM,ChenKC,etal.CalcineurinenhancesL-typeCa(2+)channelactivityinhippocampalneurons:increasedeffectwithageinculture.Neuroscience.2002;110(2):213-25.PMID:11958864.
PerrinoBA.Regulationofcalcineurinphosphataseactivitybyitsautoinhibitorydomain.ArchBiochemBiophys.1999Dec1;372(1):159-65.PMID:10562429.