Description
BI-2536isapolo-likekinase1(PLK1)inhibitorthatdisruptsmitosisandcelldivision.BI-2536exhibitsanticanceractivityandmayinduceapoptosisincancercells.
BI-2536isapolo-likekinase1(PLK1)inhibitorthatdisruptsmitosisandcelldivision.BI-2536exhibitsanticanceractivityandmayinduceapoptosisincancercells.
| CasNo. | 755038-02-9 |
|---|---|
| Purity | ≥98% |
| Formula | C28H39N7O3 |
| FormulaWt. | 521.65 |
| Synonym | BI2536 |
| Appearance | Paleyellowtooff-whitepowder |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | B3200InfoSheetPDF |
|---|
ColnaghiR,WheatleySP.LiaisonsbetweensurvivinandPlk1duringcelldivisionandcelldeath.JBiolChem.2010Jul16;285(29):22592-604.PMID:20427271.
ZhangJ,YangPL,GrayNS.Targetingcancerwithsmallmoleculekinaseinhibitors.NatureReviewsCancer.2009Jan;9:28-39.