FenoldopamisabenzazepinederivativethatactsasapartialagoNISTatD1receptors;itmayalsoinhibitα1-adrenergicreceptors.Fenoldopamexhibitsvasodilatory,antihypertensive,andnatriureticactivities.Invivo,fenoldopamdecreasesbloodpressure,afterload,andbloodflow;italsoinhibitsNaClreabsorptioninthethickascendinglimb,promotingNa+excretion.
| CasNo. | 67227-57-0 |
|---|---|
| Purity | ≥98% |
| Formula | C16H16ClNO3S•CH3SO3H |
| FormulaWt. | 401.87 |
| ChemicalName | 6-Chloro-2,3,4,5-tetrahydro-1-(4-hydroxyphenyl)-1H-3-benzazepine-7,8-diolmethanesulfonate |
| IUPACName | 9-chloro-5-(4-hydroxyphenyl)-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol;methanesulfonicacid |
| Synonym | Fenoldopammethanesulfonate;Corlopam |
| MeltingPoint | 274°C(dec) |
| Solubility | Solubleinwater.DMSO15mg/mL. |
| Appearance | Whitetooffwhitepowder |
| StoreTemp | Ambient |
|---|---|
| ShipTemp | Ambient |
| MSDS | F1654MSDSPDF |
|---|---|
| InfoSheet | F1654InfoSheetPDF |
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