CTAPisanantagoNISTatμ-opioidreceptors(μORs)thatexhibitsneuromodulatoryactivity.CTAPpreventsreinstatementofdrugseekinginanimalmodelsofethanoladdiction.CTAPalsopreventsopioid-induceddecreasesininflammatorycytokinereleaseinanimalmodelsofintestinalischemia/reperfusion.Additionally,CTAPinhibitsopioid-inducedanalgesiainanimalmodelsofcolorectaldistension.
| Purity | ≥95% |
|---|---|
| Formula | C51H67N13O11S |
| FormulaWt. | 1102.33 |
| IUPACName | (4R,7S,10S,13S,16S,19R)-N-[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]-19-[[(2S)-2-amino-3-phenylpropanoyl]amino]-10-[3-(diaminomethylideneamino)propyl]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-3,3-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | C7602InfoSheetPDF |
|---|
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