DAMGOisasyntheticpeptideμ-opioidreceptoragoNIST(μOR)thatexhibitsneuromodulatoryandantinociceptive/analgesicactivities.DAMGOdecreasespaineffectsinanimalmodelsofvisceralpainandalsodecreasesmotoractivityinseparateanimalmodels.Invitroandinvivo,DAMGOdecreaseslevelsoftheglutamatetransporterEAAT3anddecreasesGABA-Acurrent.
| Purity | ≥95% |
|---|---|
| Formula | C26H35N5O6 |
| FormulaWt. | 513.0 |
| IUPACName | (2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-1-(2-hydroxyethylamino)-1-oxo-3-phenylpropan-2-yl]-methylamino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide |
| Synonym | DAGO;DAMGE |
| Appearance | Whitetooffwhitepowder |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | D0025InfoSheetPDF |
|---|
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