Deltorphin I is an opioid peptide that acts as an agonist at δ-opioid receptors (δORs). Deltorphin I exhibits antinociceptive and pro-angiogenic activities. In vitro, deltorphin I stimulates proliferation, migration, adhesion, and tube formation.
| Cas No. | 122752-15-2 |
|---|---|
| Purity | ≥98% |
| Formula | C37H52N8O10 |
| Formula Wt. | 768.87 |
| Chemical Name | Glycinamide,L-tyrosyl-D-alanyl-L-phenylalanyl-L-alpha-aspartyl-L-valyl-L-valyl- |
| IUPAC Name | (3S)-3-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]-4-[[1-[[(2S)-1-[(2-amino-2-oxoethyl)amino]-3-methyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-4-oxobutanoic acid |
| Synonym | Deltorphin C; Deltophin 1; Deltorphin I, ala(2)-; [D-Ala2]-Deltorphin I |
| Appearance | White to off white powder |
| Store Temp | -20°C |
|---|---|
| Ship Temp | Ambient |
| Info Sheet | D1644 Info Sheet PDF |
|---|
Dai X, Song HJ, Cui SG, et al. The stimulative effects of endogenous opioids on endothelial cell proliferation, migration and angiogenesis in vitro. Eur J Pharmacol. 2010 Feb 25;628(1-3):42-50. PMID: 19932695.
Li SR, Wang T, Wang R, et al. Melatonin enhances antinociceptive effects of delta-, but not mu-opioid agonist in mice. Brain Res. 2005 May 10;1043(1-2):132-8. PMID: 15862526.
