Description
C59isaPORCNinhibitorthatexhibitsanticancerchemotherapeuticactivity,inhibitingtheprogressionofmammarytumorsinvivobydownregulatingWntsignaling.
C59isaPORCNinhibitorthatexhibitsanticancerchemotherapeuticactivity,inhibitingtheprogressionofmammarytumorsinvivobydownregulatingWntsignaling.
CasNo. | 1243243-89-1 |
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Purity | ≥98% |
Formula | C25H21N3O |
FormulaWt. | 379.45 |
IUPACName | 2-[4-(2-methylpyridin-4-yl)phenyl]-N-(4-pyridin-3-ylphenyl)acetamide |
Synonym | Wnt-C59 |
Appearance | Whitetooffwhitepowder |
StoreTemp | -20°C |
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ShipTemp | Ambient |
InfoSheet | C0800InfoSheetPDF |
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ProffittKD,MadanB,KeZ,etal.PharmacologicalinhibitionoftheWntacyltransferasePORCNpreventsgrowthofWNT-drivenmammarycancer.CancerRes.2013Jan15;73(2):502-7.PMID:23188502.