MastoparanXisanantimicrobial/antibacterialpeptide(AMP)derivedfromthevenomofbeesandwasps.MastoparanXactivatesmastcellsthroughbindingandactivationoftheGαsubunitofGPCRs.MastoparanXentersintoneutralandnegativelychargedmembranes,causingformationandleakageofgiantunilamellarvesiclesandinducingbarrierdisruptions.
| CasNo. | 72093-22-2 |
|---|---|
| Purity | ≥95% |
| Formula | C73H126N20O15S |
| FormulaWt. | 1556.01 |
| IUPACName | (2S)-N-[(2S)-1-[[(2S)-6-amino-1-[[2-[[(3S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-6-amino-1-[[(2S)-6-amino-1-[[(2S)-1-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxohexan-2-yl]amino]-1-oxopropan-2-yl]amino]-4-methylsulfanyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxohexan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-[[(2S,3S)-2-amino-3-methylpentanoyl]amino]butanediamide |
| Synonym | Mastcelldegranulatingpeptide(Vespaxanthoptera)(9CI) |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | M0173InfoSheetPDF |
|---|
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