Description
MelanostatinisaneuromodulatorypeptideoftheMIF-1family.MelanostatinmodulatesD2receptordopaminesignalinganddownstreameffects.Additionally,thispeptidepotentiatesantidepressantactivityofamitriptylineanddesipramineintheforcedswimtest.
MelanostatinisaneuromodulatorypeptideoftheMIF-1family.MelanostatinmodulatesD2receptordopaminesignalinganddownstreameffects.Additionally,thispeptidepotentiatesantidepressantactivityofamitriptylineanddesipramineintheforcedswimtest.
Purity | ≥95% |
---|---|
Formula | C189H285N53O57S |
FormulaWt. | 4243.76 |
Synonym | MIF-1 |
StoreTemp | -20°C |
---|---|
ShipTemp | Ambient |
InfoSheet | M1648InfoSheetPDF |
---|
PanW,KastinAJ.FromMIF-1toendomorphin:theTyr-MIF-1familyofpeptides.Peptides.2007Dec;28(12):2411-34.PMID:17988762.
MishraRK,MakmanMH,CostainWJ,etal.ModulationofagoNISTstimulatedadenylylcyclaseandGTPaseactivitybyL-pro-L-leu-glycinamideanditspeptidomimeticanalogueinratstriatalmembranes.NeurosciLett.1999Jul2;269(1):21-4.PMID:10821635.
KostowskiW,DanyszW,DyrW,etal.MIF-1potentiatestheactionoftricyclicantidepressantsinananimalmodelofdepression.Peptides.1991Sep-Oct;12(5):915-8.PMID:1686934.