Description
DefactinibinhibitsFAKanddisplaysanticanceractivity.Inovariancancermodels,thiscompounddecreasescellproliferation,inducesapoptosis,anddecreasestumorweight.
DefactinibinhibitsFAKanddisplaysanticanceractivity.Inovariancancermodels,thiscompounddecreasescellproliferation,inducesapoptosis,anddecreasestumorweight.
| CasNo. | 1073154-85-4 |
|---|---|
| Purity | ≥98% |
| Formula | C20H21F3N8O3S |
| FormulaWt. | 510.49 |
| Synonym | VS-6063,PF-04554878 |
| Appearance | Whitetooffwhitepowder |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | D1722InfoSheetPDF |
|---|
LeeBY,TimpsonP,HorvathLG,etal.FAKsignalinginhumancancerasatargetfortherapeutics.PharmacolTher.2015Feb;146C:132-149.PMID:25316657.
KangY,HuW,IvanC,etal.RoleoffocaladhesionkinaseinregulatingYB-1-mediatedpaclitaxelresistanceinovariancancer.JNatlCancerInst.2013Oct2;105(19):1485-95.PMID:24062525.