Description
DefactinibinhibitsFAKanddisplaysanticanceractivity.Inovariancancermodels,thiscompounddecreasescellproliferation,inducesapoptosis,anddecreasestumorweight.
DefactinibinhibitsFAKanddisplaysanticanceractivity.Inovariancancermodels,thiscompounddecreasescellproliferation,inducesapoptosis,anddecreasestumorweight.
CasNo. | 1073154-85-4 |
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Purity | ≥98% |
Formula | C20H21F3N8O3S |
FormulaWt. | 510.49 |
Synonym | VS-6063,PF-04554878 |
Appearance | Whitetooffwhitepowder |
StoreTemp | -20°C |
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ShipTemp | Ambient |
InfoSheet | D1722InfoSheetPDF |
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LeeBY,TimpsonP,HorvathLG,etal.FAKsignalinginhumancancerasatargetfortherapeutics.PharmacolTher.2015Feb;146C:132-149.PMID:25316657.
KangY,HuW,IvanC,etal.RoleoffocaladhesionkinaseinregulatingYB-1-mediatedpaclitaxelresistanceinovariancancer.JNatlCancerInst.2013Oct2;105(19):1485-95.PMID:24062525.