Description
LEE011isaninhibitorofCDK4/6thatexhibitsanticancerchemotherapeuticactivity.Inneuroblastomacells,LEE011inducescellcyclearrestandcellularsenescence,inhibitingproliferation.Inanimalmodels,LEE011inhibitstumorxenograftgrowth.
LEE011isaninhibitorofCDK4/6thatexhibitsanticancerchemotherapeuticactivity.Inneuroblastomacells,LEE011inducescellcyclearrestandcellularsenescence,inhibitingproliferation.Inanimalmodels,LEE011inhibitstumorxenograftgrowth.
| CasNo. | 1211441-98-3 |
|---|---|
| Purity | ≥98% |
| FormulaWt. | 434.54 |
| IUPACName | 7-cyclopentyl-N,N-dimethyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrrolo[2,3-d]pyrimidine-6-carboxamide |
| Synonym | LEE011,Ribociclib |
| Appearance | Off-whitePowder |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | L1616InfoSheetPDF |
|---|
RaderJ,RussellMR,HartLS,etal.DualCDK4/CDK6inhibitioninducescell-cyclearrestandsenescenceinneuroblastoma.ClinCancerRes.2013Nov15;19(22):6173-82.PMID:24045179.