Description
LEE011isaninhibitorofCDK4/6thatexhibitsanticancerchemotherapeuticactivity.Inneuroblastomacells,LEE011inducescellcyclearrestandcellularsenescence,inhibitingproliferation.Inanimalmodels,LEE011inhibitstumorxenograftgrowth.
LEE011isaninhibitorofCDK4/6thatexhibitsanticancerchemotherapeuticactivity.Inneuroblastomacells,LEE011inducescellcyclearrestandcellularsenescence,inhibitingproliferation.Inanimalmodels,LEE011inhibitstumorxenograftgrowth.
CasNo. | 1211441-98-3 |
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Purity | ≥98% |
FormulaWt. | 434.54 |
IUPACName | 7-cyclopentyl-N,N-dimethyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrrolo[2,3-d]pyrimidine-6-carboxamide |
Synonym | LEE011,Ribociclib |
Appearance | Off-whitePowder |
StoreTemp | -20°C |
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ShipTemp | Ambient |
InfoSheet | L1616InfoSheetPDF |
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RaderJ,RussellMR,HartLS,etal.DualCDK4/CDK6inhibitioninducescell-cyclearrestandsenescenceinneuroblastoma.ClinCancerRes.2013Nov15;19(22):6173-82.PMID:24045179.