Description
INCB28060isaninhibitorofc-METthatexhibitsanticancerchemotherapeuticactivity.Incellularmodelsofcancer,INCB28060inhibitscellmigrationandinducesapoptosis,inhibitingproliferation.Inanimalmodels,thiscompoundinhibitstumorgrowth.
INCB28060isaninhibitorofc-METthatexhibitsanticancerchemotherapeuticactivity.Incellularmodelsofcancer,INCB28060inhibitscellmigrationandinducesapoptosis,inhibitingproliferation.Inanimalmodels,thiscompoundinhibitstumorgrowth.
CasNo. | 1029712-80-8 |
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Purity | ≥98% |
Formula | C23H17FN6O |
FormulaWt. | 412.42 |
IUPACName | 2-fluoro-N-methyl-4-[7-(quinolin-6-ylmethyl)imidazo[1,2-b][1,2,4]triazin-2-yl]benzamide |
Synonym | INC-280,Capmatinib |
Appearance | YellowPowder |
StoreTemp | 4°C |
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ShipTemp | Ambient |
MSDS | I5208MSDSPDF |
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InfoSheet | I5208InfoSheetPDF |
LiuX,WangQ,YangG,etal.Anovelkinaseinhibitor,INCB28060,blocksc-MET-dependentsignaling,neoplasticactivities,andcross-talkwithEGFRandHER-3.ClinCancerRes.2011Nov15;17(22):7127-38.PMID:21918175.