Description
KX1-004isanindolethatinhibitsSrc.Thiscompounddecreasesapoptosisinhaircellstopreventnoise-inducedhearingloss.
KX1-004isanindolethatinhibitsSrc.Thiscompounddecreasesapoptosisinhaircellstopreventnoise-inducedhearingloss.
| CasNo. | 518058-84-9 |
|---|---|
| Purity | ≥98% |
| Formula | C16H13FN2O2 |
| FormulaWt. | 284.29 |
| IUPACName | 5-Fluoro-N-(3-hydroxybenzyl)-1H-indole-2-carboxamide |
| StoreTemp | -20°C |
|---|---|
| ShipTemp | Ambient |
| InfoSheet | K9200InfoSheetPDF |
|---|
FetoniAR,BielefeldEC,PaludettiG,etal.Aputativeroleofp53pathwayagainstimpulsenoiseinduceddamageasdemonstratedbyprotectionwithpifithrin-alphaandaSrcinhibitor.NeurosciRes.2014Apr-May;81-82:30-7.PMID:24472721.
BielefeldEC,HangauerD,HendersonD.Protectionfromimpulsenoise-inducedhearinglosswithnovelSrc-proteintyrosinekinaseinhibitors.NeurosciRes.2011Dec;71(4):348-54.PMID:21840347.
HarrisKC,HuB,HangauerD,etal.Preventionofnoise-inducedhearinglosswithSrc-PTKinhibitors.HearRes.2005Oct;208(1-2):14-25.PMID:15950415.